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New Thiazole Acetic Acid Derivatives: A Study to Screen Cardiovascular Activity Using Isolated Rat Hearts and Blood Vessels

Cardiovascular diseases are one of the major causes of mortalities worldwide. In the present research, new synthetic derivatives of thiazole were studied using isolated hearts and blood vessels of rats. The heart and thoracic aorta were tested with six new synthesized thiazole acetic acid derivative...

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Autores principales: Raghunatha, P., Inamdar, Mohammed Naseeruddin, Asdaq, Syed Mohammed Basheeruddin, Almuqbil, Mansour, Alzahrani, Abdullah R., Alaqel, Saleh I., Kamal, Mehnaz, Alsubaie, Firas Hamdan, Alsanie, Walaa F., Alamri, Abdulhakeem S., Rabbani, Syed Imam, Attimarad, Mahesh, Mohan, S., Alhomrani, Majid
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2022
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9572953/
https://www.ncbi.nlm.nih.gov/pubmed/36234675
http://dx.doi.org/10.3390/molecules27196138
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author Raghunatha, P.
Inamdar, Mohammed Naseeruddin
Asdaq, Syed Mohammed Basheeruddin
Almuqbil, Mansour
Alzahrani, Abdullah R.
Alaqel, Saleh I.
Kamal, Mehnaz
Alsubaie, Firas Hamdan
Alsanie, Walaa F.
Alamri, Abdulhakeem S.
Rabbani, Syed Imam
Attimarad, Mahesh
Mohan, S.
Alhomrani, Majid
author_facet Raghunatha, P.
Inamdar, Mohammed Naseeruddin
Asdaq, Syed Mohammed Basheeruddin
Almuqbil, Mansour
Alzahrani, Abdullah R.
Alaqel, Saleh I.
Kamal, Mehnaz
Alsubaie, Firas Hamdan
Alsanie, Walaa F.
Alamri, Abdulhakeem S.
Rabbani, Syed Imam
Attimarad, Mahesh
Mohan, S.
Alhomrani, Majid
author_sort Raghunatha, P.
collection PubMed
description Cardiovascular diseases are one of the major causes of mortalities worldwide. In the present research, new synthetic derivatives of thiazole were studied using isolated hearts and blood vessels of rats. The heart and thoracic aorta were tested with six new synthesized thiazole acetic acid derivatives (SMVA-10, SMVA-35, SMVA-40, SMVA-41, SMVA-42 and SMVA-60), and the data obtained were statistically analyzed and compared. Isolated rat hearts were used to record the changes in developed tension and heart rate, while thoracic aortas were used to measure the contractile response, before and after treatments. Analysis of the results indicated a significant (p < 0.01) increase in developed tension with the addition of SMVA-35, SMVA-40, SMVA-41 and SMVA-42, which was augmented in the presence of adrenaline without affecting the heart rate. On the other hand, acetylcholine significantly decreased the developed tension, which was significantly reversed (p < 0.01) in the presence of compounds (SMVA-35 and SMVA-60). However, in the presence of SMVA-35 and SMVA-40, acetylcholine-induced bradycardia was significantly (p < 0.01) reduced. Furthermore, only SMVA-42 induced a dose-dependent contractile response in the isolated blood vessel, which was abolished in the presence of prazosin. Therefore, it can be concluded that some of the new synthesized thiazole derivatives exhibited promising results by raising the developed tension without changing the heart rate or blood vessel function, which could be helpful in failing heart conditions. However, more research is required to fully comprehend the function, mechanism and effectiveness of the compounds.
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spelling pubmed-95729532022-10-17 New Thiazole Acetic Acid Derivatives: A Study to Screen Cardiovascular Activity Using Isolated Rat Hearts and Blood Vessels Raghunatha, P. Inamdar, Mohammed Naseeruddin Asdaq, Syed Mohammed Basheeruddin Almuqbil, Mansour Alzahrani, Abdullah R. Alaqel, Saleh I. Kamal, Mehnaz Alsubaie, Firas Hamdan Alsanie, Walaa F. Alamri, Abdulhakeem S. Rabbani, Syed Imam Attimarad, Mahesh Mohan, S. Alhomrani, Majid Molecules Article Cardiovascular diseases are one of the major causes of mortalities worldwide. In the present research, new synthetic derivatives of thiazole were studied using isolated hearts and blood vessels of rats. The heart and thoracic aorta were tested with six new synthesized thiazole acetic acid derivatives (SMVA-10, SMVA-35, SMVA-40, SMVA-41, SMVA-42 and SMVA-60), and the data obtained were statistically analyzed and compared. Isolated rat hearts were used to record the changes in developed tension and heart rate, while thoracic aortas were used to measure the contractile response, before and after treatments. Analysis of the results indicated a significant (p < 0.01) increase in developed tension with the addition of SMVA-35, SMVA-40, SMVA-41 and SMVA-42, which was augmented in the presence of adrenaline without affecting the heart rate. On the other hand, acetylcholine significantly decreased the developed tension, which was significantly reversed (p < 0.01) in the presence of compounds (SMVA-35 and SMVA-60). However, in the presence of SMVA-35 and SMVA-40, acetylcholine-induced bradycardia was significantly (p < 0.01) reduced. Furthermore, only SMVA-42 induced a dose-dependent contractile response in the isolated blood vessel, which was abolished in the presence of prazosin. Therefore, it can be concluded that some of the new synthesized thiazole derivatives exhibited promising results by raising the developed tension without changing the heart rate or blood vessel function, which could be helpful in failing heart conditions. However, more research is required to fully comprehend the function, mechanism and effectiveness of the compounds. MDPI 2022-09-20 /pmc/articles/PMC9572953/ /pubmed/36234675 http://dx.doi.org/10.3390/molecules27196138 Text en © 2022 by the authors. https://creativecommons.org/licenses/by/4.0/Licensee MDPI, Basel, Switzerland. This article is an open access article distributed under the terms and conditions of the Creative Commons Attribution (CC BY) license (https://creativecommons.org/licenses/by/4.0/).
spellingShingle Article
Raghunatha, P.
Inamdar, Mohammed Naseeruddin
Asdaq, Syed Mohammed Basheeruddin
Almuqbil, Mansour
Alzahrani, Abdullah R.
Alaqel, Saleh I.
Kamal, Mehnaz
Alsubaie, Firas Hamdan
Alsanie, Walaa F.
Alamri, Abdulhakeem S.
Rabbani, Syed Imam
Attimarad, Mahesh
Mohan, S.
Alhomrani, Majid
New Thiazole Acetic Acid Derivatives: A Study to Screen Cardiovascular Activity Using Isolated Rat Hearts and Blood Vessels
title New Thiazole Acetic Acid Derivatives: A Study to Screen Cardiovascular Activity Using Isolated Rat Hearts and Blood Vessels
title_full New Thiazole Acetic Acid Derivatives: A Study to Screen Cardiovascular Activity Using Isolated Rat Hearts and Blood Vessels
title_fullStr New Thiazole Acetic Acid Derivatives: A Study to Screen Cardiovascular Activity Using Isolated Rat Hearts and Blood Vessels
title_full_unstemmed New Thiazole Acetic Acid Derivatives: A Study to Screen Cardiovascular Activity Using Isolated Rat Hearts and Blood Vessels
title_short New Thiazole Acetic Acid Derivatives: A Study to Screen Cardiovascular Activity Using Isolated Rat Hearts and Blood Vessels
title_sort new thiazole acetic acid derivatives: a study to screen cardiovascular activity using isolated rat hearts and blood vessels
topic Article
url https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9572953/
https://www.ncbi.nlm.nih.gov/pubmed/36234675
http://dx.doi.org/10.3390/molecules27196138
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