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Design and synthesis of some new benzoylthioureido benzenesulfonamide derivatives and their analogues as carbonic anhydrase inhibitors
The present investigation reports the design and synthesis of three series of benzoylthioureido derivatives bearing either benzenesulfonamide 7a–f, benzoic acid 8a–f or ethylbenzoate 9a–f moieties. The synthesised compounds were screened for their carbonic anhydrase inhibitory activity (CAI) against...
Autores principales: | Oudah, Khulood H., Mahmoud, Walaa R., Awadallah, Fadi M., Taher, Azza T., Abbas, Safinaz E.-S, Allam, Heba Abdelrasheed, Vullo, Daniela, Supuran, Claudiu T. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Taylor & Francis
2022
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9621292/ https://www.ncbi.nlm.nih.gov/pubmed/36305274 http://dx.doi.org/10.1080/14756366.2022.2132485 |
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