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3H-1,2-Benzoxaphosphepine 2-oxides as selective inhibitors of carbonic anhydrase IX and XII

The synthesis of 3H-1,2-benzoxaphosphepine 2-oxides and evaluation of their inhibitory activity against human carbonic anhydrase (hCA) isoforms I, II, IX, and XII are described. The target compounds were obtained via a concise synthesis from commercial salicylaldehydes and displayed low to sub-micro...

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Detalles Bibliográficos
Autores principales:	Pustenko, Aleksandrs, Balašova, Anastasija, Nocentini, Alessio, Supuran, Claudiu T., Žalubovskis, Raivis
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Taylor & Francis 2022
Materias:	Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9668280/ https://www.ncbi.nlm.nih.gov/pubmed/36377338 http://dx.doi.org/10.1080/14756366.2022.2143496

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