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Privileged Scaffold Decoration for the Identification of the First Trisubstituted Triazine with Anti-SARS-CoV-2 Activity
Current therapy against severe acute respiratory syndrome coronavirus type 2 (SARS-CoV-2) are based on the use of Remdesivir 1, Molnupiravir 2, and the recently identified Nirmatrelvir 3. Unfortunately, these three drugs showed some limitations regarding potency and possible drug–drug interactions....
Autores principales: | Cesarini, Silvia, Vicenti, Ilaria, Poggialini, Federica, Secchi, Massimiliano, Giammarino, Federica, Varasi, Ilenia, Lodola, Camilla, Zazzi, Maurizio, Dreassi, Elena, Maga, Giovanni, Botta, Lorenzo, Saladino, Raffaele |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2022
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9782877/ https://www.ncbi.nlm.nih.gov/pubmed/36557962 http://dx.doi.org/10.3390/molecules27248829 |
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