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Convenient Synthesis of N-Heterocycle-Fused Tetrahydro-1,4-diazepinones

A general approach towards the synthesis of tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-4-one, tetrahydro[1,4]diazepino[1,2-a]indol-1-one and tetrahydro-1H-benzo[4,5]imidazo[1,2-a][1,4]diazepin-1-one derivatives was introduced. A regioselective strategy was developed for synthesizing ethyl 1-(oxiran-...

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Detalles Bibliográficos
Autores principales:	Dzedulionytė, Karolina, Veikšaitė, Melita, Morávek, Vít, Malinauskienė, Vida, Račkauskienė, Greta, Šačkus, Algirdas, Žukauskaitė, Asta, Arbačiauskienė, Eglė
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2022
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9783606/ https://www.ncbi.nlm.nih.gov/pubmed/36557800 http://dx.doi.org/10.3390/molecules27248666

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