Cargando…

Diarylation of thiazolopyrimidines by laccase and their in vitro evaluation as antitumor agents

A mild and efficient method was developed for the synthesis of new derivatives of thiazolo[3,2-a] pyrimidin-3(2H)-ones from available starting materials based on the oxidation of catechols to ortho-quinone by Myceliophthora thermophila laccase (Novozym 51,003) and 1,4-addition of active methylene ca...

Descripción completa

Detalles Bibliográficos
Autores principales:	Shahedi, Mansour, Shahani, Rojina, Habibi, Zohreh, Yousefi, Maryam, Brask, Jesper, Minaei-Tehrani, Arash, Samadi, Fatemeh Yazdi, Mohammadi, Mehdi
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Nature Publishing Group UK 2022
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9790884/ https://www.ncbi.nlm.nih.gov/pubmed/36567332 http://dx.doi.org/10.1038/s41598-022-26820-9

Ejemplares similares

Biocatalytic decarboxylative Michael addition for synthesis of 1,4-benzoxazinone derivatives
por: Bavandi, Hossein, et al.
Publicado: (2022)

Immobilization of Thermomyces lanuginosus lipase through isocyanide-based multi component reaction on multi-walled carbon nanotube: application for kinetic resolution of rac-ibuprofen
por: Moguei, Mohamad Reza Safarpoor, et al.
Publicado: (2022)

Thiazolopyrimidine derivatives as novel class of small molecule tyrosinase inhibitor
por: Ghasemi, Nastaran, et al.
Publicado: (2023)

Identification of the Allosteric Binding Site for Thiazolopyrimidine on the C-Type Lectin Langerin
por: Zhang, Hengxi, et al.
Publicado: (2022)

Chitosan nanoparticle loaded by epidermal growth factor as a potential protein carrier for wound healing: In vitro and in vivo studies
por: Montazeri, Samaneh, et al.
Publicado: (2023)

Microwave assisted synthesis of some new thiazolopyrimidine and pyrimidothiazolopyrimidopyrimidine derivatives with potential antimicrobial activity
por: Youssef, Ayman M. S., et al.
Publicado: (2018)

Synthesis and Cytotoxic Activity of New Thiazolopyrimidine Sugar Hydrazones and Their Derived Acyclic Nucleoside Analogues
por: Basiony, Ebtesam A., et al.
Publicado: (2020)

Microwave Assisted Synthesis of Some New Thiazolopyrimidine, Thiazolodipyrimidine and Thiazolopyrimidothiazolopyrimidine Derivatives with Potential Antioxidant and Antimicrobial Activity
por: Youssef, Mohamed M., et al.
Publicado: (2012)

Photoinduced synthesis of unsymmetrical diaryl selenides from triarylbismuthines and diaryl diselenides
por: Kobiki, Yohsuke, et al.
Publicado: (2013)

Combined experimental and TD-DFT/DMOl(3) investigations, optical properties, and photoluminescence behavior of a thiazolopyrimidine derivative
por: Abozeed, Amina A., et al.
Publicado: (2022)

Vicinal Diaryl-Substituted Isoxazole and Pyrazole Derivatives with In Vitro Growth Inhibitory and In Vivo Antitumor Activity
por: Turanlı, Sümeyye, et al.
Publicado: (2022)

Homocouplings of Sodium Arenesulfinates: Selective Access to Symmetric Diaryl Sulfides and Diaryl Disulfides
por: Yu, Xin-Zhang, et al.
Publicado: (2022)

Discovery of Hybrid Dual N-Acylhydrazone and Diaryl Urea Derivatives as Potent Antitumor Agents: Design, Synthesis and Cytotoxicity Evaluation
por: Zhai, Xin, et al.
Publicado: (2013)

Hydroxide-Mediated S(N)Ar Rearrangement for Synthesis of Novel Depside Derivatives Containing Diaryl Ether Skeleton as Antitumor Agents
por: Yu, Xiang, et al.
Publicado: (2023)

Synthesis and Anticancer Activity of New 1-Thia-4-azaspiro[4.5]decane, Their Derived Thiazolopyrimidine and 1,3,4-Thiadiazole Thioglycosides
por: Flefel, Eman M., et al.
Publicado: (2017)

Laccase purified from Cerrena unicolor exerts antitumor activity against leukemic cells
por: MATUSZEWSKA, ANNA, et al.
Publicado: (2016)

Photo-Inactivation of Staphylococcus aureus by Diaryl-Porphyrins
por: Orlandi, Viviana Teresa, et al.
Publicado: (2023)

Synthesis and Antiproliferative Activity of Steroidal Diaryl Ethers
por: Kovács, Édua, et al.
Publicado: (2023)

Iodine-Mediated Oxidative Rearrangement of α,β-Unsaturated Diaryl Ketones: A Facile Access to 1,2-Diaryl Diketones
por: Bansode, Ajay H., et al.
Publicado: (2019)

Design and Synthesis of Fluorescent 1,3-Diaryl-β-carbolines and 1,3-Diaryl-3,4-dihydro-β-carbolines
por: Pu, JiYang, et al.
Publicado: (2021)

Magnetic mesocellular foams with nickel complexes: as efficient and reusable nanocatalysts for the synthesis of symmetrical and asymmetrical diaryl chalcogenides
por: Shirvandi, Zeinab, et al.
Publicado: (2022)

Synthesis of Novel Benzodifuranyl; 1,3,5-Triazines; 1,3,5-Oxadiazepines; and Thiazolopyrimidines Derived from Visnaginone and Khellinone as Anti-Inflammatory and Analgesic Agents
por: Abu-Hashem, Ameen Ali, et al.
Publicado: (2020)

Design, Synthesis, and Bioevaluation of Indole Core Containing 2-Arylidine Derivatives of Thiazolopyrimidine as Multitarget Inhibitors of Cholinesterases and Monoamine Oxidase A/B for the Treatment of Alzheimer Disease
por: Shahid Nadeem, Muhammad, et al.
Publicado: (2022)

Stable Radical Cations of N,N′‐Diarylated Dihydrodiazapentacenes
por: Xie, Gaozhan, et al.
Publicado: (2019)

Stable N,N’‐Diarylated Dihydrodiazaacene Radical Cations
por: Xie, Gaozhan, et al.
Publicado: (2020)

Photoinactivation of Pseudomonas aeruginosa Biofilm by Dicationic Diaryl-Porphyrin
por: Orlandi, Viviana Teresa, et al.
Publicado: (2021)

Diaryl-Pyrano-Chromenes Atropisomers: Stereodynamics and Conformational Studies
por: Ciogli, Alessia, et al.
Publicado: (2023)

Multiple Reaction Monitoring for quantitative laccase kinetics by LC-MS
por: Perna, Valentina, et al.
Publicado: (2018)

Screening of ligands for the Ullmann synthesis of electron-rich diaryl ethers
por: Otto, Nicola, et al.
Publicado: (2012)

Palladium-Catalyzed Oxidative Regio- and Diastereoselective Diarylating Carbocyclization of Dienynes
por: Jiang, Min, et al.
Publicado: (2013)

Diaryl Disulfides as Novel Stabilizers of Tumor Suppressor Pdcd4
por: Schmid, Tobias, et al.
Publicado: (2016)

Inhibition of Leishmania infantum trypanothione reductase by diaryl sulfide derivatives
por: Saccoliti, Francesco, et al.
Publicado: (2017)

TDAE Strategy for the Synthesis of 2,3-Diaryl N-Tosylaziridines
por: Khoumeri, Omar, et al.
Publicado: (2013)

Identification of Diaryl-Quinoline Compounds as Entry Inhibitors of Ebola Virus
por: Cui, Qinghua, et al.
Publicado: (2018)

Oxidative Rearrangement of Stilbenes to 2,2-Diaryl-2-hydroxyacetaldehydes
por: Kalshetti, Rupali G., et al.
Publicado: (2020)

Synthesis of Diaryl Hydroxyl Dicarboxylic Acids from Amino Acids
por: Eronen, Aleksi E.K., et al.
Publicado: (2020)

Clarification on the Reactivity of Diaryl Diselenides toward Hexacyclohexyldilead under Light
por: Hung, Vu Thai, et al.
Publicado: (2021)

A one-pot cascade protocol for diarylation of amines and water
por: Linde, Erika, et al.
Publicado: (2022)

Copper-promoted S-arylation reactions with triarylbismuths for the synthesis of diaryl sulfides
por: Nie, Mei, et al.
Publicado: (2023)

Advanced Synthesis of Conductive Polyaniline Using Laccase as Biocatalyst
por: de Salas, Felipe, et al.
Publicado: (2016)

Cannot write session to /tmp/vufind_sessions/sess_stnlc8dureqdtl4mit554a58q2