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Indole Derivatives as New Structural Class of Potent and Antiproliferative Inhibitors of Monocarboxylate Transporter 1 (MCT1; SLC16A1)

[Image: see text] The solute carrier (SLC) monocarboxylate transporter 1 (MCT1; SLC16A1) represents a promising target for the treatment of cancer; however, the MCT1 modulator landscape is underexplored with only roughly 100 reported compounds. To expand the knowledge about MCT1 modulation, we synth...

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Detalles Bibliográficos
Autores principales:	Puri, Sachin, Stefan, Katja, Khan, Sharuk L., Pahnke, Jens, Stefan, Sven Marcel, Juvale, Kapil
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2022
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9841531/ https://www.ncbi.nlm.nih.gov/pubmed/36584238 http://dx.doi.org/10.1021/acs.jmedchem.2c01612

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