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Novel thiazolone-benzenesulphonamide inhibitors of human and bacterial carbonic anhydrases

A small library of novel thiazolone-benzenesulphonamides has been prepared and evaluated for their ability to inhibit three human cytosolic carbonic anhydrases (hCA I, hCA II, and hCA VII) and three bacterial carbonic anhydrases (MscCAβ, StCA1, and StCA2). All investigated hCAs were inhibited by the...

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Detalles Bibliográficos
Autores principales:	Abdoli, Morteza, De Luca, Viviana, Capasso, Clemente, Supuran, Claudiu T., Žalubovskis, Raivis
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Taylor & Francis 2023
Materias:	Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9848287/ https://www.ncbi.nlm.nih.gov/pubmed/36629426 http://dx.doi.org/10.1080/14756366.2022.2163243

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