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Monocarbonyl Curcumin Analogues as Potent Inhibitors against Human Glutathione Transferase P1-1

The isoenzyme of human glutathione transferase P1-1 (hGSTP1-1) is involved in multi-drug resistance (MDR) mechanisms in numerous cancer cell lines. In the present study, the inhibition potency of two curcuminoids and eleven monocarbonyl curcumin analogues against hGSTP1-1 was investigated. Demethoxy...

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Detalles Bibliográficos
Autores principales:	Pantiora, Panagiota, Furlan, Veronika, Matiadis, Dimitris, Mavroidi, Barbara, Perperopoulou, Fereniki, Papageorgiou, Anastassios C., Sagnou, Marina, Bren, Urban, Pelecanou, Maria, Labrou, Nikolaos E.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2022
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9854774/ https://www.ncbi.nlm.nih.gov/pubmed/36670925 http://dx.doi.org/10.3390/antiox12010063

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