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Rationalizing the Binding Modes of PET Radiotracers Targeting the Norepinephrine Transporter

Purpose: A new PET radiotracer (18)F-AF78 showing great potential for clinical application has been reported recently. It belongs to a new generation of phenethylguanidine-based norepinephrine transporter (NET)-targeting radiotracers. Although many efforts have been made to develop NET inhibitors as...

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Detalles Bibliográficos
Autores principales:	Tutov, Anna, Chen, Xinyu, Werner, Rudolf A., Mühlig, Saskia, Zimmermann, Thomas, Nose, Naoko, Koshino, Kazuhiro, Lapa, Constantin, Decker, Michael, Higuchi, Takahiro
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2023
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9963373/ https://www.ncbi.nlm.nih.gov/pubmed/36840011 http://dx.doi.org/10.3390/pharmaceutics15020690

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