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Synthesis and radiolabelling of PSMA-targeted derivatives containing GYK/MVK cleavable linkers

Targeted radionuclide therapy (TRT) is a promising strategy to treat different types of cancer. TRT relies on a targeting vector used to deliver a therapeutic radionuclide specifically to the tumour site. Several low molecular weight ligands targeting the prostate-specific membrane antigen (PSMA) ha...

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Detalles Bibliográficos
Autores principales:	Murce, Erika, de Blois, Erik, van den Berg, Sophie, de Jong, Marion, Seimbille, Yann
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	The Royal Society 2023
Materias:	Chemistry
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9993039/ https://www.ncbi.nlm.nih.gov/pubmed/36908985 http://dx.doi.org/10.1098/rsos.220950

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