Mostrando 1 - 20 Resultados de 43,917 Para Buscar '"antagonist"', tiempo de consulta: 0.63s Limitar resultados
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    “…In this article, we will explore the scientific and clinical case for an ACTH antagonist, and will review the evidence for existing and recently described peptides and modified peptides in this role.…”
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    “…Hydroxymethylthiohydantoin, hydroxymethylthiohydantoin, and hydantoin, containing a pyridine group, were synthesized to study their androgen receptor antagonistic activities. Among them, compounds 6a/6c/7g/19a/19b exhibited excellent androgen receptor antagonistic activity, which was consistent with or even superior to enzalutamide. …”
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    “…The role of the two receptors has been delineated using highly selective ET(A) (BQ123, TAK-044) and ET(B) (BQ788) peptide antagonists. Nonpeptide antagonists, bosentan, macitentan, and ambrisentan, that are either mixed ET(A)/ET(B) antagonists or display ET(A) selectivity, have been approved for clinical use but to date are limited to pulmonary hypertension. …”
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    por Doods, H. N., Schindler, M.
    Publicado 2001
    “…The presentation will focus on BIBN 4096 BS, since this compound is still the only potent calcitonin gene-related peptide (CGRP)-antagonist described so far[1].…”
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    por Bubna, Aditya Kumar
    Publicado 2021
    “…Leukotriene antagonists constitute an important group of drugs in the therapeutic armamentarium of all dermatologists. …”
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    por Lochner, Martin, Thompson, Andrew J.
    Publicado 2016
    “…Scopolamine is a high affinity muscarinic antagonist that is used for the prevention of post-operative nausea and vomiting. 5-HT(3) receptor antagonists are used for the same purpose and are structurally related to scopolamine. …”
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    “…The present study investigated the effects of intraperitoneal (IP) injection of cannabinoid CB1 receptor antagonist (AM251) in the presence of alpha-1 adrenergic antagonist (Prazosin) on rat behavior in the EPM. …”
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    por Yocum, David
    Publicado 2004
    “…Tumor necrosis factor (TNF) antagonists are biologic response modifiers that have significantly improved functional outcomes in patients with rheumatoid arthritis (RA). …”
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    por Oh, Yun Kyu
    Publicado 2008
    “…Several non-peptide vasopressin receptor antagonists have been developed and are being studied primarily for treating conditions characterized by hyponatremia and fluid overload. …”
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    por Watanabe, Masaki, Kakuta, Hiroki
    Publicado 2018
    “…Retinoid X receptor (RXR) antagonists are not only useful as chemical tools for biological research, but are also candidate drugs for the treatment of various diseases, including diabetes and allergies, although no RXR antagonist has yet been approved for clinical use. …”
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    “…A comprehensive review of pharmacological and medical aspects of the muscarinic class of acetylcholine agonists and antagonists is presented. The therapeutic benefits of achieving receptor subtype selectivity are outlined and applications in the treatment of Alzheimer’s disease are discussed. …”
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