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Inhibition of Acid-Sensing Ion Channels by KB-R7943, a Reverse Na(+)/Ca(2+) Exchanger Inhibitor

KB-R7943, an isothiourea derivative, is widely used as a pharmacological inhibitor of reverse sodium–calcium exchanger (NCX). It has been shown to have neuroprotective and analgesic effects in animal models; however, the detailed molecular mechanisms remain elusive. In the current study, we investig...

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Detalles Bibliográficos
Autores principales:	Sun, Hua-Wei, Chu, Xiang-Ping, Simon, Roger P., Xiong, Zhi-Gang, Leng, Tian-Dong
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2023
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10046550/ https://www.ncbi.nlm.nih.gov/pubmed/36979442 http://dx.doi.org/10.3390/biom13030507

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