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Synthesis, radiolabeling, and evaluation of 68Ga-labeled aminoquinoxaline derivative as a potent PFKFB3-targeted PET tracer

Glycolysis, as a multi-step oxidation process, plays important roles in the energy supply for living cells, including malignant tumor cells. Recent studies have revealed that 6-phosphofructo-2-kinase/fructose-2,6-biphosphatase 3 (named PFKFB3), a bifunctional enzyme in glycolysis, is upregulated in...

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Detalles Bibliográficos
Autores principales: Chen, Feng, Wu, Yi, Ma, Yixuan, Yin, Honghai, Su, Feijing, Huang, Rui, Wu, Xiaoai, Liu, Qian
Formato: Online Artículo Texto
Lenguaje:English
Publicado: Frontiers Media S.A. 2023
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10073729/
https://www.ncbi.nlm.nih.gov/pubmed/37035116
http://dx.doi.org/10.3389/fchem.2023.1158503