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Styrylquinazoline derivatives as ABL inhibitors selective for different DFG orientations
Among tyrosine kinase inhibitors, quinazoline-based compounds represent a large and well-known group of multi-target agents. Our previous studies have shown interesting kinases inhibition activity for a series of 4-aminostyrylquinazolines based on the CP-31398 scaffold. Here, we synthesised a new se...
Autores principales: | Malarz, Katarzyna, Mularski, Jacek, Pacholczyk, Marcin, Musiol, Robert |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Taylor & Francis
2023
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10120462/ https://www.ncbi.nlm.nih.gov/pubmed/37070569 http://dx.doi.org/10.1080/14756366.2023.2201410 |
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