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Cytotoxic Activity of α-Aminophosphonic Derivatives Coming from the Tandem Kabachnik–Fields Reaction and Acylation

Encouraged by the significant cytotoxic activity of simple α-aminophosphonates, a molecular library comprising phosphonoylmethyl- and phosphinoylmethyl-α-aminophosphonates, a tris derivative, and N-acylated species was established. The promising aminophosphonate derivatives were subjected to a compa...

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Detalles Bibliográficos
Autores principales: Varga, Petra R., Szabó, Rita Oláhné, Dormán, György, Bősze, Szilvia, Keglevich, György
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2023
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10144033/
https://www.ncbi.nlm.nih.gov/pubmed/37111263
http://dx.doi.org/10.3390/ph16040506