Distinct Profiles of Desensitization of µ-Opioid Receptors Caused by Remifentanil or Fentanyl: In Vitro Assay with Cells and Three-Dimensional Structural Analyses

Remifentanil (REM) and fentanyl (FEN) are commonly used analgesics that act by activating a µ-opioid receptor (MOR). Although optimal concentrations of REM can be easily maintained during surgery, it is sometimes switched to FEN for optimal pain regulation. However, standards for this switching prot...

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Detalles Bibliográficos
Autores principales: Uezono, Eiko, Mizobuchi, Yusuke, Miyano, Kanako, Ohbuchi, Katsuya, Murata, Hiroaki, Komatsu, Akane, Manabe, Sei, Nonaka, Miki, Hirokawa, Takatsugu, Yamaguchi, Keisuke, Iseki, Masako, Uezono, Yasuhito, Hayashida, Masakazu, Kawagoe, Izumi
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2023
Materias:
Article
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10179353/
https://www.ncbi.nlm.nih.gov/pubmed/37176075
http://dx.doi.org/10.3390/ijms24098369

Internet

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10179353/
https://www.ncbi.nlm.nih.gov/pubmed/37176075
http://dx.doi.org/10.3390/ijms24098369

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