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Site-Selective C–H Amination of Phenol-Containing Biomolecules

[Image: see text] A C–N bond-forming cross-dehydrogenative coupling of a collection of Tyr-containing peptides and estrogens with heteroarenes is described. This oxidative coupling is distinguished by its scalability, operational simplicity, and air tolerance and enables the appendance of phenothiaz...

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Detalles Bibliográficos
Autores principales: Girón-Elola, Carlota, Sasiain, Ibon, Sánchez-Fernández, Rosalía, Pazos, Elena, Correa, Arkaitz
Formato: Online Artículo Texto
Lenguaje:English
Publicado: American Chemical Society 2023
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10278169/
https://www.ncbi.nlm.nih.gov/pubmed/37284781
http://dx.doi.org/10.1021/acs.orglett.3c01560