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Synthesis of Benzocycloalkanone-Based Michael Acceptors and Biological Activities as Antimalarial and Antitrypanosomal Agents

A series of benzocycloalkanone derivatives have been prepared and evaluated as antimalarial and antitrypanosomal agents. The compounds were obtained by direct coupling of preformed 4-substituted benzaldehyde and indanone or tetralone substitutes through aldol condensation of Claisen-Schmidt using so...

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Detalles Bibliográficos
Autores principales:	Mijoba, Ali, Fernandez-Moreira, Esteban, Parra-Giménez, Nereida, Espinosa-Tapia, Sandra, Blanco, Zuleyma, Ramírez, Hegira, Charris, Jaime E.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2023
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10385825/ https://www.ncbi.nlm.nih.gov/pubmed/37513441 http://dx.doi.org/10.3390/molecules28145569

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