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Benzenesulfonamide Analogs: Synthesis, Anti-GBM Activity and Pharmacoprofiling

The tropomyosin receptor kinase A (TrkA) family of receptor tyrosine kinases (RTKs) emerge as a potential target for glioblastoma (GBM) treatment. Benzenesulfonamide analogs were identified as kinase inhibitors possessing promising anticancer properties. In the present work, four known and two novel...

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Detalles Bibliográficos
Autores principales: Murugesan, Akshaya, Konda Mani, Saravanan, Thiyagarajan, Ramesh, Palanivel, Suresh, Gurbanov, Atash V., Zubkov, Fedor I., Kandhavelu, Meenakshisundaram
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2023
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10418358/
https://www.ncbi.nlm.nih.gov/pubmed/37569654
http://dx.doi.org/10.3390/ijms241512276