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Metabotropic Glutamate Receptor Subtype 5 Positron-Emission-Tomography Radioligands as a Tool for Central Nervous System Drug Development: Between Progress and Setbacks

The metabotropic glutamate receptor subtype 5 (mGluR5) is a class C G-protein-coupled receptor (GPCR) that has been implicated in various neuronal processes and, consequently, in several neuropsychiatric or neurodevelopmental disorders. Over the past few decades, mGluR5 has become a major focus for...

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Detalles Bibliográficos
Autores principales: Dupont, Anne-Claire, Arlicot, Nicolas, Vercouillie, Johnny, Serrière, Sophie, Maia, Serge, Bonnet-Brilhault, Frédérique, Santiago-Ribeiro, Maria-Joao
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2023
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10458693/
https://www.ncbi.nlm.nih.gov/pubmed/37631042
http://dx.doi.org/10.3390/ph16081127