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Inhibitory Mechanism of Quercimeritrin as a Novel α-Glucosidase Selective Inhibitor

In this study, 12 flavonoid glycosides were selected based on virtual screening and the literature, and Quercimeritrin was selected as the best selective inhibitor of α-glucosidase through in vitro enzyme activity inhibition experiments. Its IC(50) value for α-glucosidase was 79.88 µM, and its IC(50...

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Detalles Bibliográficos
Autores principales: Guo, Fengyu, An, Jie, Wang, Minlong, Zhang, Weibo, Chen, Chong, Mao, Xueying, Liu, Siyuan, Wang, Pengjie, Ren, Fazheng
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2023
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10528180/
https://www.ncbi.nlm.nih.gov/pubmed/37761124
http://dx.doi.org/10.3390/foods12183415