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EGFR and PI3K/m-TOR inhibitors: design, microwave assisted synthesis and anticancer activity of thiazole–coumarin hybrids

A series of thiazoline and thiazolidinone-based 4-hydroxycoumarin derivatives were synthesized using both conventional synthesis procedures and microwave-assisted techniques. The new compounds were evaluated for their cytotoxic effect against three human cancer cell lines; MCF-7, HCT-116 and HepG2 a...

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Detalles Bibliográficos
Autores principales:	Batran, Rasha Z., Ahmed, Eman Y., Awad, Hanem M., Ali, Korany A., Abdel Latif, Nehad A.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	The Royal Society of Chemistry 2023
Materias:	Chemistry
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10548181/ https://www.ncbi.nlm.nih.gov/pubmed/37800132 http://dx.doi.org/10.1039/d3ra03483f

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