Cargando…

Structural insights into the agonists binding and receptor selectivity of human histamine H(4) receptor

Histamine is a biogenic amine that participates in allergic and inflammatory processes by stimulating histamine receptors. The histamine H(4) receptor (H(4)R) is a potential therapeutic target for chronic inflammatory diseases such as asthma and atopic dermatitis. Here, we show the cryo-electron mic...

Descripción completa

Detalles Bibliográficos
Autores principales: Im, Dohyun, Kishikawa, Jun-ichi, Shiimura, Yuki, Hisano, Hiromi, Ito, Akane, Fujita-Fujiharu, Yoko, Sugita, Yukihiko, Noda, Takeshi, Kato, Takayuki, Asada, Hidetsugu, Iwata, So
Formato: Online Artículo Texto
Lenguaje:English
Publicado: Nature Publishing Group UK 2023
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10589313/
https://www.ncbi.nlm.nih.gov/pubmed/37863901
http://dx.doi.org/10.1038/s41467-023-42260-z