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Macrocyclic Peptides Closed by a Thioether–Bipyridyl Unit That Grants Cell Membrane Permeability
[Image: see text] Membrane permeability is an important factor that determines the virtue of peptides targeting intracellular molecules. By introducing a membrane penetration motif, some peptides exhibit better membrane permeabilities. Previous choices for such motifs have usually been polycationic...
Autores principales: | Chen, Hongxue, Katoh, Takayuki, Suga, Hiroaki |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
American Chemical Society
2023
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Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10591297/ https://www.ncbi.nlm.nih.gov/pubmed/37876498 http://dx.doi.org/10.1021/acsbiomedchemau.3c00027 |
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