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Synthesis and vectorial functionalisation of pyrazolo[3,4-c]pyridines

Heterocycles are a cornerstone of fragment-based drug discovery (FBDD) due to their prevalence in biologically active compounds. However, novel heterocyclic fragments are only valuable if they can be suitably elaborated to compliment a chosen target protein. Here we describe the synthesis of 5-halo-...

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Detalles Bibliográficos
Autores principales:	Bedwell, Elizabeth V., da Silva Emery, Flavio, Clososki, Giuliano C., Steel, Patrick G.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	The Royal Society of Chemistry 2023
Materias:	Chemistry
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10667592/ https://www.ncbi.nlm.nih.gov/pubmed/38024964 http://dx.doi.org/10.1039/d3ra07458g

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