Cargando…
In Vivo Evaluation of α7 Nicotinic Acetylcholine Receptor Agonists [(11)C]A-582941 and [(11)C]A-844606 in Mice and Conscious Monkeys
BACKGROUND: The α7 nicotinic acetylcholine receptors (nAChRs) play an important role in the pathophysiology of neuropsychiatric diseases such as schizophrenia and Alzheimer's disease. The goal of this study was to evaluate the two carbon-11-labeled α7 nAChR agonists [(11)C]A-582941 and [(11)C]A...
Autores principales: | Toyohara, Jun, Ishiwata, Kiichi, Sakata, Muneyuki, Wu, Jin, Nishiyama, Shingo, Tsukada, Hideo, Hashimoto, Kenji |
---|---|
Formato: | Texto |
Lenguaje: | English |
Publicado: |
Public Library of Science
2010
|
Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC2813863/ https://www.ncbi.nlm.nih.gov/pubmed/20126539 http://dx.doi.org/10.1371/journal.pone.0008961 |
Ejemplares similares
-
Occupancy of α7 Nicotinic Acetylcholine Receptors in the Brain by Tropisetron: A Positron Emission Tomography Study Using [(11)C]CHIBA-1001 in Healthy Human Subjects
por: Ishikawa, Masatomo, et al.
Publicado: (2011) -
[(11)C]CHIBA-1001 as a Novel PET Ligand for α7 Nicotinic Receptors in the Brain: A PET Study in Conscious Monkeys
por: Hashimoto, Kenji, et al.
Publicado: (2008) -
Age-Related Decrease in Male Extra-Striatal Adenosine A(1) Receptors Measured Using
(11)C-MPDX PET
por: Mishina, Masahiro, et al.
Publicado: (2017) -
Synthesis and evaluation of N-isopropyl-p-[(11)C]methylamphetamine as a novel cerebral blood flow tracer for positron emission tomography
por: Toyohara, Jun, et al.
Publicado: (2020) -
Assessment of safety, efficacy, and dosimetry of a novel 18-kDa translocator protein ligand, [(11)C]CB184, in healthy human volunteers
por: Sakata, Muneyuki, et al.
Publicado: (2017)