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Investigation of the Structure Requirement for 5-HT(6) Binding Affinity of Arylsulfonyl Derivatives: A Computational Study
5-HT(6) receptor has been implicated in a series of diseases including anxiety, depression, schizophrenia and cognitive dysfunctions. 5-HT(6) ligands have been reported to play a significant role in the treatment for central nervous system (CNS) diseases. Presently, a large series of 223 5-HT(6) lig...
Autores principales: | , , , |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Molecular Diversity Preservation International (MDPI)
2011
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3179148/ https://www.ncbi.nlm.nih.gov/pubmed/21954341 http://dx.doi.org/10.3390/ijms12085011 |