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Investigation of the Structure Requirement for 5-HT(6) Binding Affinity of Arylsulfonyl Derivatives: A Computational Study

5-HT(6) receptor has been implicated in a series of diseases including anxiety, depression, schizophrenia and cognitive dysfunctions. 5-HT(6) ligands have been reported to play a significant role in the treatment for central nervous system (CNS) diseases. Presently, a large series of 223 5-HT(6) lig...

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Detalles Bibliográficos
Autores principales: Hao, Ming, Li, Yan, Li, Hanqing, Zhang, Shuwei
Formato: Online Artículo Texto
Lenguaje:English
Publicado: Molecular Diversity Preservation International (MDPI) 2011
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3179148/
https://www.ncbi.nlm.nih.gov/pubmed/21954341
http://dx.doi.org/10.3390/ijms12085011