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2,3-Dihydro-1H-cyclopenta[b]quinoline Derivatives as Acetylcholinesterase Inhibitors—Synthesis, Radiolabeling and Biodistribution
In the present study we describe the synthesis and biological assessment of new tacrine analogs in the course of inhibition of acetylcholinesterase. The obtained molecules were synthesized in a condensation reaction between activated 6-BOC-hydrazinopyridine-3-carboxylic acid and 8-aminoalkyl derivat...
Autores principales: | Szymański, Paweł, Lázničková, Alice, Lázniček, Milan, Bajda, Marek, Malawska, Barbara, Markowicz, Magdalena, Mikiciuk-Olasik, Elżbieta |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Molecular Diversity Preservation International (MDPI)
2012
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3431846/ https://www.ncbi.nlm.nih.gov/pubmed/22949848 http://dx.doi.org/10.3390/ijms130810067 |
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