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N-Amino-imidazolin-2-one Peptide Mimic Synthesis and Conformational Analysis

[Image: see text] Base-promoted 5-exo-dig cyclizations of aza-propargylglycinamides provided N-amino-imidazolin-2-one peptide mimics, which exhibited turn geometry in X-ray crystallographic and NMR spectroscopic analyses. Sonogashira coupling prior to cyclization afforded N-amino-imidazolin-2-ones w...

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Detalles Bibliográficos
Autores principales:	Proulx, Caroline, Lubell, William D.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2012
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3437692/ https://www.ncbi.nlm.nih.gov/pubmed/22892053 http://dx.doi.org/10.1021/ol302021n

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