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Synthesis and biological activity of N-substituted-tetrahydro-γ-carbolines containing peptide residues
The synthesis of novel peptide conjugates of N-substituted-tetrahydro-γ-carbolines has been performed using the sequence of the Ugi multicomponent reaction and Cu(I)-catalyzed click chemistry. The effect of obtained γ-carboline–peptide conjugates on the rat liver mitochondria was evaluated. It was f...
Autores principales: | Sokolova, Nadezhda V, Nenajdenko, Valentine G, Sokolov, Vladimir B, Vinogradova, Daria V, Shevtsova, Elena F, Dubova, Ludmila G, Bachurin, Sergey O |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Beilstein-Institut
2014
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3896248/ https://www.ncbi.nlm.nih.gov/pubmed/24454569 http://dx.doi.org/10.3762/bjoc.10.13 |
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