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Identification of Novel Serotonin Transporter Compounds by Virtual Screening
[Image: see text] The serotonin (5-hydroxytryptamine, 5-HT) transporter (SERT) plays an essential role in the termination of serotonergic neurotransmission by removing 5-HT from the synaptic cleft into the presynaptic neuron. It is also of pharmacological importance being targeted by antidepressants...
Autores principales: | Gabrielsen, Mari, Kurczab, Rafał, Siwek, Agata, Wolak, Małgorzata, Ravna, Aina W., Kristiansen, Kurt, Kufareva, Irina, Abagyan, Ruben, Nowak, Gabriel, Chilmonczyk, Zdzisław, Sylte, Ingebrigt, Bojarski, Andrzej J. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
American Chemical
Society
2014
|
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3982395/ https://www.ncbi.nlm.nih.gov/pubmed/24521202 http://dx.doi.org/10.1021/ci400742s |
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