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Design, Synthesis and Biological Evaluation of Tasiamide Analogues as Tumor Inhibitors

Eighteen analogues of the marine cytotoxic linear peptide tasiamide were designed, synthesized and screened for their inhibitory activities against the growth of human nasopharyngeal carcinoma (KB) and human non-small cell lung tumor (A549) cell lines. The results indicated that minor modifications...

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Detalles Bibliográficos
Autores principales:	Zhang, Wei, Sun, Tiantian, Ma, Zhenhua, Li, Yingxia
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2014
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4012464/ https://www.ncbi.nlm.nih.gov/pubmed/24759000 http://dx.doi.org/10.3390/md12042308

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