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Esters of valerenic acid as potential prodrugs
Valerenic acid (VA) is a β(2/3) subunit-specific modulator of γ-aminobutyric acid (GABA) type A (GABA(A)) receptors inducing anxiolysis. Here we analyze if VA-esters can serve as prodrugs and if different ester structures have different in vitro/in vivo effects. Modulation of GABA(A) receptors expre...
Autores principales: | , , , , , , , , |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Elsevier Science
2014
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4062961/ https://www.ncbi.nlm.nih.gov/pubmed/24680924 http://dx.doi.org/10.1016/j.ejphar.2014.03.019 |