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Synthesis and antibacterial activities of acylide derivatives bearing an aryl-tetrazolyl chain

Seventeen acylides bearing an aryl-tetrazolyl alkyl-substituted side chain were synthesized, starting from clarithromycin, via several reactions including hydrolysis, acetylating, esterification, carbamylation, and Michael addition. The structures of all new compounds were confirmed by (1)H nuclear...

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Detalles Bibliográficos
Autores principales:	Shan, Ling-Xing, Sun, Ping-Hua, Guo, Bao-Qin, Xu, Xing-Jun, Li, Zhi-Qiang, Sun, Jia-Zhi, Zhou, Shu-Feng, Chen, Wei-Min
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Dove Medical Press 2014
Materias:	Original Research
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4181547/ https://www.ncbi.nlm.nih.gov/pubmed/25284984 http://dx.doi.org/10.2147/DDDT.S65673

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