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C7-Derivatization of C3-Alkylindoles Including Tryptophans and Tryptamines

[Image: see text] A versatile strategy for C7-selective boronation of tryptophans, tryptamines, and 3-alkylindoles by way of a single-pot C2/C7-diboronation–C2-protodeboronation sequence is described. The combination of a mild iridium-catalyzed C2/C7-diboronation followed by an in situ palladium-cat...

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Detalles Bibliográficos
Autores principales: Loach, Richard P., Fenton, Owen S., Amaike, Kazuma, Siegel, Dustin S., Ozkal, Erhan, Movassaghi, Mohammad
Formato: Online Artículo Texto
Lenguaje:English
Publicado: American Chemical Society 2014
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4241164/
https://www.ncbi.nlm.nih.gov/pubmed/25343326
http://dx.doi.org/10.1021/jo502062z