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C7-Derivatization of C3-Alkylindoles Including Tryptophans and Tryptamines
[Image: see text] A versatile strategy for C7-selective boronation of tryptophans, tryptamines, and 3-alkylindoles by way of a single-pot C2/C7-diboronation–C2-protodeboronation sequence is described. The combination of a mild iridium-catalyzed C2/C7-diboronation followed by an in situ palladium-cat...
Autores principales: | Loach, Richard P., Fenton, Owen S., Amaike, Kazuma, Siegel, Dustin S., Ozkal, Erhan, Movassaghi, Mohammad |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
American Chemical Society
2014
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Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4241164/ https://www.ncbi.nlm.nih.gov/pubmed/25343326 http://dx.doi.org/10.1021/jo502062z |
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