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Molecular Basis for Small Molecule Inhibition of G Protein-Coupled Receptor Kinases
[Image: see text] Small molecules that inhibit the protein kinase A, G, and C (AGC) family of serine/threonine kinases can exert profound effects on cell homeostasis and thereby regulate fundamental processes such as heart rate, blood pressure, and metabolism, but there is not yet a clinically appro...
Autores principales: | Homan, Kristoff T., Tesmer, John J. G. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
American Chemical
Society
2014
|
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4301174/ https://www.ncbi.nlm.nih.gov/pubmed/24984143 http://dx.doi.org/10.1021/cb5003976 |
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