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Zinc Mediated Azide–Alkyne Ligation to 1,5- and 1,4,5-Substituted 1,2,3-Triazoles

[Image: see text] A mild method for regioselective formation of 1,5-substituted 1,2,3-triazoles is described. The zinc-mediated reaction works at room temperature and is successful across a wide range of azido/alkynyl substrates. Additionally, the triazole 4-position can be further functionalized th...

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Detalles Bibliográficos
Autores principales:	Smith, Christopher D., Greaney, Michael F.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2013
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4331842/ https://www.ncbi.nlm.nih.gov/pubmed/24001177 http://dx.doi.org/10.1021/ol402225d

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