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Preclinical to Clinical Translation of CNS Transporter Occupancy of TD-9855, a Novel Norepinephrine and Serotonin Reuptake Inhibitor
BACKGROUND: Monoamine reuptake inhibitors exhibit unique clinical profiles that reflect distinct engagement of the central nervous system (CNS) transporters. METHODS: We used a translational strategy, including rodent pharmacokinetic/pharmacodynamic modeling and positron emission tomography (PET) im...
Autores principales: | Smith, Jacqueline AM, Patil, DL, Daniels, OT, Ding, Y-S, Gallezot, J-D, Henry, S, Kim, KHS, Kshirsagar, S, Martin, WJ, Obedencio, GP, Stangeland, E, Tsuruda, PR, Williams, W, Carson, RE, Patil, ST |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Oxford University Press
2015
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4368888/ https://www.ncbi.nlm.nih.gov/pubmed/25522383 http://dx.doi.org/10.1093/ijnp/pyu027 |
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