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The facile construction of the phthalazin-1(2H)-one scaffold via copper-mediated C–H(sp(2))/C–H(sp) coupling under mild conditions

A novel strategy for the construction of the phthalazin-1(2H)-one scaffold has been developed by means of a copper-mediated cascade C–H/C–H coupling and intramolecular annulations and a subsequent facile hydrazinolysis. This C–H activation transformation proceeds smoothly with wide generality, good...

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Detalles Bibliográficos
Autores principales:	Zhu, Wei, Wang, Bao, Zhou, Shengbin, Liu, Hong
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Beilstein-Institut 2015
Materias:	Full Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4660935/ https://www.ncbi.nlm.nih.gov/pubmed/26664581 http://dx.doi.org/10.3762/bjoc.11.177

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