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Contact-facilitated drug delivery with Sn2 lipase labile prodrugs optimize targeted lipid nanoparticle drug delivery

Sn2 lipase labile phospholipid prodrugs in conjunction with contact-facilitated drug delivery offer an important advancement in Nanomedicine. Many drugs incorporated into nanosystems, targeted or not, are substantially lost during circulation to the target. However, favorably altering the pharmacoki...

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Detalles Bibliográficos
Autores principales: Pan, Dipanjan, Pham, Christine TN, Weilbaecher, Katherine N, Tomasson, Michael H, Wickline, Samuel A, Lanza, Gregory M
Formato: Online Artículo Texto
Lenguaje:English
Publicado: John Wiley & Sons, Inc. 2016
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4709477/
https://www.ncbi.nlm.nih.gov/pubmed/26296541
http://dx.doi.org/10.1002/wnan.1355