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Virtual Screening of DrugBank Reveals Two Drugs as New BCRP Inhibitors

The breast cancer resistance protein (BCRP) is an ABC transporter playing a crucial role in the pharmacokinetics of drugs. The early identification of substrates and inhibitors of this efflux transporter can help to prevent or foresee drug-drug interactions. In this work, we built a ligand-based in...

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Detalles Bibliográficos
Autores principales:	Montanari, Floriane, Cseke, Anna, Wlcek, Katrin, Ecker, Gerhard F.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	SAGE Publications 2016
Materias:	Original Research
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5302078/ https://www.ncbi.nlm.nih.gov/pubmed/27401583 http://dx.doi.org/10.1177/1087057116657513

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