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Peptides with 6-Aminohexanoic Acid: Synthesis and Evaluation as Plasmin Inhibitors
Fifteen new peptide derivatives of ɛ-aminocaproic acid (EACA) containing the known fragment –Ala–Phe–Lys– with an affinity for plasmin were synthesised in the present study. The synthesis was carried out a solid phase. The following compounds were synthesised: H–Phe–Lys–EACA–X, H–d-Ala–Phe–Lys–EACA–...
Autores principales: | Purwin, Maciej, Markowska, Agnieszka, Bruzgo, Irena, Rusak, Tomasz, Surażyński, Arkadiusz, Jaworowska, Urszula, Midura-Nowaczek, Krystyna |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Springer Netherlands
2016
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5401710/ https://www.ncbi.nlm.nih.gov/pubmed/28491013 http://dx.doi.org/10.1007/s10989-016-9555-3 |
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