Cargando…

Facile one-pot four-component synthesis of 3,4-dihydro-2-pyridone derivatives: novel urease inhibitor scaffold

In the current study, a series of 3,4-dihydro-2-pyridone derivatives were synthesized in a one-pot fourcomponent reaction of Meldrum's acid, benzaldehyde derivatives, methyl acetoacetate, and ammonium acetate. SiO2-Pr-SO3H was used as an efficient catalyst for the synthesis of the target compou...

Descripción completa

Detalles Bibliográficos
Autores principales:	Hakimi, Arash Modarres, Lashgari, Negar, Mahernia, Shabnam, Ziarani, Ghodsi Mohammadi, Amanlou, Massoud
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Medknow Publications & Media Pvt Ltd 2017
Materias:	Original Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5615865/ https://www.ncbi.nlm.nih.gov/pubmed/28974973 http://dx.doi.org/10.4103/1735-5362.213980

Ejemplares similares

Urease Inhibitory Activities of some Commonly Consumed Herbal Medicines
por: Mahernia, Shabnam, et al.
Publicado: (2015)

Green Synthesis and Urease Inhibitory Activity of Spiro-Pyrimidinethiones/Spiro-Pyrimidinones-Barbituric Acid Derivatives
por: Mohammadi Ziarani, Ghodsi, et al.
Publicado: (2015)

Synthesis of Some Spiro Indeno[1,2-b]pyrido[2,3-d]Pyrimidine-5,3′-Indolines as New Urease Inhibitors
por: Mohammadi Ziarani, Ghodsi, et al.
Publicado: (2016)

Three-component synthesis of pyrano[2,3-d]-pyrimidine dione derivatives facilitated by sulfonic acid nanoporous silica (SBA-Pr-SO(3)H) and their docking and urease inhibitory activity
por: Ziarani, Ghodsi Mohammadi, et al.
Publicado: (2013)

Determination of hydrogen cyanide concentration in mainstream smoke of tobacco products by polarography
por: Mahernia, Shabnam, et al.
Publicado: (2015)

Recent advances in the application of indoles in multicomponent reactions
por: Mohammadi Ziarani, Ghodsi, et al.
Publicado: (2018)

The role of hollow magnetic nanoparticles in drug delivery
por: Mohammadi Ziarani, Ghodsi, et al.
Publicado: (2019)

Efficient Synthesis and Antimicrobial Evaluation of Pyrazolopyranopyrimidines in the Presence of SBA-Pr-SO3H as a Nanoporous Acid Catalyst
por: Mohammadi Ziarani, Ghodsi, et al.
Publicado: (2018)

3,4-Dihydro-2(1H)-Pyridones as Building Blocks of Synthetic Relevance
por: Chalán-Gualán, Sisa, et al.
Publicado: (2022)

Infrared Assisted Production of 3,4-Dihydro-2(1H)-pyridones in Solvent-Free Conditions
por: Noguez, M. Olivia, et al.
Publicado: (2011)

Effects of onopordia, a novel isolated compound from Onopordon acanthium, on pentylenetetrazole-induced seizures in mice: Possible involvement of nitric oxide pathway
por: Hassanzadeh, Malihe, et al.
Publicado: (2019)

Screening of 20 Commonly Used Iranian Traditional Medicinal Plants Against Urease
por: Biglar, Mahmood, et al.
Publicado: (2014)

Recent advances on the synthesis of natural pyrrolizidine alkaloids: alexine, and its stereoisomers
por: Mohammadi Ziarani, Ghodsi, et al.
Publicado: (2022)

Urease inhibitory activities of β-boswellic acid derivatives
por: Golbabaei, Sanaz, et al.
Publicado: (2013)

Prediction of new Hsp90 inhibitors based on 3,4-isoxazolediamide scaffold using QSAR study, molecular docking and molecular dynamic simulation
por: Abbasi, Maryam, et al.
Publicado: (2017)

Large scale screening of commonly used Iranian traditional medicinal plants against urease activity
por: Nabati, Farzaneh, et al.
Publicado: (2012)

A Preliminary Investigation of the Jack-Bean Urease Inhibition by Randomly Selected Traditionally Used Herbal Medicine
por: Biglar, Mahmood, et al.
Publicado: (2012)

Arylmethylene hydrazine derivatives containing 1,3-dimethylbarbituric moiety as novel urease inhibitors
por: Pedrood, Keyvan, et al.
Publicado: (2021)

Design and synthesis of new N-thioacylated ciprofloxacin derivatives as urease inhibitors with potential antibacterial activity
por: Pedrood, Keyvan, et al.
Publicado: (2022)

Isoindolin-1-ones Fused to Barbiturates: From Design and Molecular Docking to Synthesis and Urease Inhibitory Evaluation
por: Kazemzadeh, Houman, et al.
Publicado: (2022)

An efficient and ecofriendly synthesis of highly functionalized pyridones via a one-pot three-component reaction
por: Hosseini, Hajar, et al.
Publicado: (2018)

Tankyrase Inhibitor for Cardiac Tissue Regeneration: an In-silico Approach
por: Hosseini, Faezeh Sadat, et al.
Publicado: (2021)

New advances on Au–magnetic organic hybrid core–shells in MRI, CT imaging, and drug delivery
por: Mohajer, Fatemeh, et al.
Publicado: (2021)

Exploration of Thiourea-Based Scaffolds for the Construction of Bacterial Ureases Inhibitors
por: Tabor, Wojciech, et al.
Publicado: (2023)

Synthesis of 4-Pyridone-3-sulfate and an improved synthesis of 3-Hydroxy-4-Pyridone
por: Behrman, Edward J
Publicado: (2009)

Design and synthesis of novel nitrothiazolacetamide conjugated to different thioquinazolinone derivatives as anti-urease agents
por: Sohrabi, Marzieh, et al.
Publicado: (2022)

5-Methyl-2-pyridone
por: Mao, Shulin, et al.
Publicado: (2011)

2-Pyridone: monoclinic polymorph
por: Arman, Hadi D., et al.
Publicado: (2009)

Rational design of yolk–shell nanostructures for drug delivery
por: Mohammadi Ziarani, Ghodsi, et al.
Publicado: (2020)

Applications of SBA-15 supported Pd metal catalysts as nanoreactors in C–C coupling reactions
por: Mohammadi Ziarani, Ghodsi, et al.
Publicado: (2018)

New thioxothiazolidinyl-acetamides derivatives as potent urease inhibitors: design, synthesis, in vitro inhibition, and molecular dynamic simulation
por: Dastyafteh, Navid, et al.
Publicado: (2023)

Flavonoids and related privileged scaffolds as potential urease inhibitors: a review
por: Al-Rooqi, Munirah M., et al.
Publicado: (2023)

Facile One-Pot Synthesis of Functionalized Quinoline-Fused Fluorescent Dihydro/Spiro-quinazolinone Derivatives
por: George, Kevin, et al.
Publicado: (2022)

N-Aryl-3,4-dihydroisoquinoline Carbothioamide Analogues as Potential Urease Inhibitors
por: Ali, Fayaz, et al.
Publicado: (2021)

Acenaphtoquinoxaline as a selective fluorescent sensor for Hg (II) detection: experimental and theoretical studies
por: Darroudi, Mahdieh, et al.
Publicado: (2020)

A preliminary investigation of anticholinesterase activity of some Iranian medicinal plants commonly used in traditional medicine
por: Jazayeri, Seyed Behzad, et al.
Publicado: (2014)

One-pot two-step catalytic synthesis of 6-amino-2-pyridone-3,5-dicarbonitriles enabling anti-cancer bioactivity
por: Nicely, Lynden G., et al.
Publicado: (2022)

The Biochemical Pathways of Nicotinamide-Derived Pyridones
por: Hayat, Faisal, et al.
Publicado: (2021)

(3-Nitrophenyl)methanediyl diacetate
por: Mohammadi Ziarani, Ghodsi, et al.
Publicado: (2007)

SBA-Pr-Is-TAP Functionalized Nanostructured Silica as a Highly Selective Fluorescent Chemosensor for Fe(3+) and Cr(2)O(7)(2−) Ions in Aqueous Media
por: Ziarani, Ghodsi Mohammadi, et al.
Publicado: (2021)

Cannot write session to /tmp/vufind_sessions/sess_qqbddu4b4289i2ks9me483sbec