Highly selective acylation of polyamines and aminoglycosides by 5-acyl-5-phenyl-1,5-dihydro-4H-pyrazol-4-ones

5-Acyl-5-phenyl-1,5-dihydro-4H-pyrazol-4-ones, accessible from arylpropargyl phenyldiazoacetates, are highly selective acyl transfer reagents for di- and polyamines, as well as aminoalcohols and aminothiols. As reagents with a carbon-based leaving group, they have been applied for benzoyl transfer w...

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Detalles Bibliográficos
Autores principales: Marichev, Kostiantyn O., Garcia, Estevan C., Bhowmick, Kartick C., Wherritt, Daniel J., Arman, Hadi, Doyle, Michael P.
Formato: Online Artículo Texto
Lenguaje:English
Publicado: Royal Society of Chemistry 2017
Materias:
Chemistry
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5635523/
https://www.ncbi.nlm.nih.gov/pubmed/29081946
http://dx.doi.org/10.1039/c7sc03184j

Internet

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5635523/
https://www.ncbi.nlm.nih.gov/pubmed/29081946
http://dx.doi.org/10.1039/c7sc03184j

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