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Synthesis of Novel C-2- or C-15-Labeled BODIPY—Estrone Conjugates

Novel BODIPY–estrone conjugates were synthesized via Cu(I)-catalyzed azide–alkyne cycloaddition (CuAAC). Estrone-alkynes or an estrone-azide as starting compounds were synthesized via Michael addition or Sonogashira reaction as key steps. Fluorescent dyes based on BODIPY-core were provided by azide...

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Detalles Bibliográficos
Autores principales:	Bacsa, Ildikó, Konc, Csilla, Orosz, Anna Boglárka, Kecskeméti, Gábor, Rigó, Réka, Özvegy-Laczka, Csilla, Mernyák, Erzsébet
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2018
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6017578/ https://www.ncbi.nlm.nih.gov/pubmed/29614041 http://dx.doi.org/10.3390/molecules23040821

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