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The discovery of pyridinium 1,2,4-triazines with enhanced performance in bioconjugation reactions
1,2,4-Triazines have recently been identified as versatile dienes participating in the inverse electron-demand Diels–Alder reaction with strained dienophiles. However, their widespread utility in bioconjugation reactions is still limited. Herein, we report a systematic study on the reactivity of var...
Autores principales: | Siegl, Sebastian J., Dzijak, Rastislav, Vázquez, Arcadio, Pohl, Radek, Vrabel, Milan |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Royal Society of Chemistry
2017
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6092722/ https://www.ncbi.nlm.nih.gov/pubmed/30155204 http://dx.doi.org/10.1039/c6sc05442k |
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