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NOP receptor pharmacological profile – A dynamic mass redistribution study
The Nociceptin/Orphanin FQ (N/OFQ) peptide NOP receptor is coupled to pertussis toxin (PTX)-sensitive G proteins (G(i/o)) whose activation leads to the inhibition of both cAMP production and calcium channel activity, and to the stimulation of potassium currents. The label free dynamic mass redistrib...
Autores principales: | Malfacini, Davide, Simon, Katharina, Trapella, Claudio, Guerrini, Remo, Zaveri, Nurulain T., Kostenis, Evi, Calo’, Girolamo |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Public Library of Science
2018
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6117024/ https://www.ncbi.nlm.nih.gov/pubmed/30161182 http://dx.doi.org/10.1371/journal.pone.0203021 |
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