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Versatility of 7-Substituted Coumarin Molecules as Antimycobacterial Agents, Neuronal Enzyme Inhibitors and Neuroprotective Agents
A medium-throughput screen using Mycobacterium tuberculosis H37Rv was employed to screen an in-house library of structurally diverse compounds for antimycobacterial activity. In this initial screen, eleven 7-substituted coumarin derivatives with confirmed monoamine oxidase-B and cholinesterase inhib...
Autores principales: | Kapp, Erika, Visser, Hanri, Sampson, Samantha L., Malan, Sarel F., Streicher, Elizabeth M., Foka, Germaine B., Warner, Digby F., Omoruyi, Sylvester I., Enogieru, Adaze B., Ekpo, Okobi E., Zindo, Frank T., Joubert, Jacques |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2017
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6151660/ https://www.ncbi.nlm.nih.gov/pubmed/28973990 http://dx.doi.org/10.3390/molecules22101644 |
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